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1

Trends in twin pregnancies and mode of delivery during the last 30 years: inconsistency between guidelines and clinical practice

Antsaklis, Aris, Malamas, Fotodotis M., Sindos, Michael

Journal:

Journal of Perinatal Medicine

Year:

2013

Language:

english

File:

PDF, 9.45 MB

english, 2013

2

Clinical pharmacology of celecoxib, a COX-2 selective inhibitor

Antoniou, Katerina, Malamas, Michael, Drosos, Alexandros A

Journal:

Expert Opinion on Pharmacotherapy

Year:

2007

Language:

english

File:

PDF, 237 KB

english, 2007

3

Inhibition of N-acylethanolamine acid amidase reduces nicotine-induced dopamine activation and reward

Sagheddu, Claudia, Scherma, Maria, Congiu, Mauro, Fadda, Paola, Carta, Gianfranca, Banni, Sebastiano, Wood, JodiAnne T., Makriyannis, Alexandros, Malamas, Michael S., Pistis, Marco

Journal:

Neuropharmacology

Year:

2019

Language:

english

File:

PDF, 717 KB

english, 2019

4

Di-substituted pyridinyl aminohydantoins as potent and highly selective human β-secretase (BACE1) inhibitors

Michael S. Malamas, Keith Barnes, Matthew Johnson, Yu Hui, Ping Zhou, Jim Turner, Yun Hu, Erik Wagner, Kristi Fan, Rajiv Chopra, Andrea Olland, Jonathan Bard, Menelas Pangalos, Peter Reinhart, Albert

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 576 KB

english, 2010

5

Preparation, reactivity, and spectral properties of 1,3-dioxin vinylogous esters: versatile .beta.-ketovinyl cation equivalents

Smith, Amos B., Dorsey, Bruce D., Ohba, Masashi, Lupo, Andrew T., Malamas, Michael S.

Journal:

Journal of Organic Chemistry

Year:

1988

Language:

english

File:

PDF, 1.56 MB

english, 1988

6

ChemInform Abstract: Design and Synthesis of Aminohydantoins (I) as Potent and Selective Human β-Secretase (BACE1) Inhibitors with Enhanced Brain Permeability.

Michael S. Malamas, et al. et al.

Journal:

Year:

2011

File:

PDF, 25 KB

2011

7

Evaluation of fluorescence-based thermal shift assays for hit identification in drug discovery

Mei-Chu Lo, Ann Aulabaugh, Guixian Jin, Rebecca Cowling, Jonathan Bard, Michael Malamas, George Ellestad

Journal:

Analytical Biochemistry

Year:

2004

Language:

english

File:

PDF, 369 KB

english, 2004

8

2,4-thiazolidinediones as potent and selective human β3 agonists

Baihua Hu, John Ellingboe, Iwan Gunawan, Stella Han, Elwood Largis, Zenan Li, Michael Malamas, Ruth Mulvey, Alexander Oliphant, Fuk-Wah Sum, Jeff Tillett, Victoria Wong

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 149 KB

english, 2001

9

Comparison of the therapeutic effects of two vanadium complexes administered at low doses on benzo[a]pyrene-induced malignant tumors in rats

Angelos Evangelou, Spiros Karkabounas, George Kalpouzos, Michael Malamas, Roman Liasko, Dimitris Stefanou, Antonis T. Vlahos, Themistoklis A. Kabanos

Journal:

Year:

1997

Language:

english

File:

PDF, 477 KB

english, 1997

10

P2-481: Small molecule BACE-1 inhibitors are potent, selective and orally active

Malamas, Michael, Erdei, Jim, Gunawan, Iwan, Robichaud, Albert, Turner, Jim, Hu, Yun, Wagner, Erik, Aschmies, Suzan, Comery, Tom, Fan, Kristi, Chopra, Rajiv, Magolda, Ron, Pangalos, Menelas, Reinhart,

Journal:

Alzheimer's & Dementia

Year:

2008

Language:

english

File:

PDF, 61 KB

english, 2008

11

Design and synthesis of cyanamides as potent and selective N-acylethanolamine acid amidase inhibitors

Malamas, Michael S., Farah, Shrouq I., Manjunath, Lamani, Pelekoudas, Dimitrios N., Thomas Perry, Nicholas, Rajarshi, Girija, Yume Miyabe, Christina, Chandrashekhar, Honrao, West, Jay, Pavlopoulos, Sp

Journal:

Bioorganic & Medicinal Chemistry

Year:

2019

Language:

english

File:

PDF, 3.22 MB

english, 2019

12

Design and Synthesis of 5,5′-Disubstituted Aminohydantoins as Potent and Selective Human β-Secretase (BACE1) Inhibitors

Malamas, Michael S., Erdei, Jim, Gunawan, Iwan, Turner, Jim, Hu, Yun, Wagner, Erik, Fan, Kristi, Chopra, Rajiv, Olland, Andrea, Bard, Jonathan, Jacobsen, Steve, Magolda, Ronald L., Pangalos, Menelas,

Journal:

Journal of Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 2.63 MB

english, 2010

13

Pyridinyl aminohydantoins as small molecule BACE1 inhibitors

Ping Zhou, Yanfang Li, Yi Fan, Zheng Wang, Rajiv Chopra, Andrea Olland, Yun Hu, Ronald L. Magolda, Menelas Pangalos, Peter H. Reinhart, M. James Turner, Jonathan Bard, Michael S. Malamas, Albert J. Ro

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 440 KB

english, 2010

14

Acylguanidine inhibitors of β-secretase: Optimization of the pyrrole ring substituents extending into the substrate binding pocket

Lee D. Jennings, Derek C. Cole, Joseph R. Stock, Mohani N. Sukhdeo, John W. Ellingboe, Rebecca Cowling, Guixian Jin, Eric S. Manas, Kristi Y. Fan, Michael S. Malamas, Boyd L. Harrison, Steve Jacobsen,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2008

Language:

english

File:

PDF, 230 KB

english, 2008

15

Investigation of the critical amino acids in the BACE1 binding site that interact with small molecule inhibitors using a novel radioligand and X-ray crystallography

Hirst, Warren D., Kubek, Katie, Bard, Jonathan, Turner, James, Fan, Kristi, Malamas, Michael, Reinhart, Peter H., Robichaud, Albert J.

Journal:

Alzheimer's & Dementia

Year:

2009

Language:

english

File:

PDF, 45 KB

english, 2009

16

Design and synthesis of aminohydantoins as potent and selective human β-secretase (BACE1) inhibitors with enhanced brain permeability

Michael S. Malamas, Albert Robichaud, Jim Erdei, Dominick Quagliato, William Solvibile, Ping Zhou, Koi Morris, Jim Turner, Erik Wagner, Kristi Fan, Andrea Olland, Steve Jacobsen, Peter Reinhart, David

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 819 KB

english, 2010

17

Discovery and initial optimization of 5,5′-disubstituted aminohydantoins as potent β-secretase (BACE1) inhibitors

Pawel Nowak, Derek C. Cole, Ann Aulabaugh, Jonathan Bard, Rajiv Chopra, Rebecca Cowling, Kristi Y. Fan, Baihua Hu, Steve Jacobsen, Minakshi Jani, Guixan Jin, Mei-Chu Lo, Michael S. Malamas, Eric S. Ma

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2010

Language:

english

File:

PDF, 593 KB

english, 2010

18

N-Substituted Spirosuccinimide, Spiropyridazine, Spiroazetidine, and Acetic Acid Aldose Reductase Inhibitors Derived from Isoquinoline-1,3-diones. 2

Malamas, Michael S., Hohman, Thomas C.

Journal:

Journal of Medicinal Chemistry

Year:

1994

Language:

english

File:

PDF, 1.46 MB

english, 1994

19

Oximes short-acting CB1 receptor agonists

Malamas, Michael S., Raghav, Jimit Girish, Ma, Xiaoy, Honrao, Chandrashekhar, Wood, JodiAnne T., Benchama, Othman, Zhou, Han, Mallipeddi, Srikrishnan, Makriyannis, Alexandros

Journal:

Bioorganic & Medicinal Chemistry

Year:

2018

Language:

english

File:

PDF, 1.76 MB

english, 2018

20

Synthesis of Heterocycle Substituted 1-Aryl-4-piperidones

Hu, Baihua, Malamas, Michael, Ellingboe, John

Journal:

Year:

2002

Language:

english

File:

PDF, 89 KB

english, 2002

21

The novel cannabinoid 1 receptor agonist AM11101 increases food intake in female rats.

Ogden, Sean B., Malamas, Michael S., Makriyannis, Alexandros, Eckel, Lisa A.

Journal:

British Journal of Pharmacology

Year:

2019

File:

PDF, 1.49 MB

2019

22

Structure-Based Design of Estrogen Receptor-β Selective Ligands

Manas, Eric S., Unwalla, Rayomand J., Xu, Zhang B., Malamas, Michael S., Miller, Chris P., Harris, Heather A., Hsiao, Chulai, Akopian, Tatos, Hum, Wah-Tung, Malakian, Karl, Wolfrom, Scott, Bapat, Asho

Journal:

Journal of the American Chemical Society

Year:

2004

Language:

english

File:

PDF, 1.18 MB

english, 2004

23

Synthesis and evaluation of potent and selective MGL inhibitors as a glaucoma treatment

Alapafuja, Shakiru O., Malamas, Michael S., Shukla, Vidya, Zvonok, Alexander, Miller, Sally, Daily, Laura, Rajarshi, Girija, Miyabe, Christina Yume, Chandrashekhar, Honrao, Wood, JodiAnne, Tyukhtenko,

Journal:

Bioorganic & Medicinal Chemistry

Year:

2018

Language:

english

File:

PDF, 1.13 MB

english, 2018

24

ChemInform Abstract: Novel Pyrrolyl 2-Aminopyridines as Potent and Selective Human β-Secretase (BACE1) Inhibitors.

Michael S. Malamas, et al. et al.

Journal:

Year:

2010

File:

PDF, 19 KB

2010

25

New oxadiazolidinedione derivatives as potent and selective human β3 agonists

Baihua Hu, Michael Malamas, John Ellingboe, Elwood Largis, Stella Han, Ruth Mulvey, Jeff Tillett

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2001

Language:

english

File:

PDF, 163 KB

english, 2001

26

Epidemiological Aspects of the Use of Cannabis among University Students in Greece

Marselos, Marios, Boutsouris, Konstantinos, Liapi, Helen, Malamas, Michael, Kateri, Maria, Papaioannou, Takis

Journal:

European Addiction Research

Year:

1997

Language:

english

File:

PDF, 1.24 MB

english, 1997

27

Metabolic Profiling of a CB2 Agonist, AM9338, Using LC-MS and Microcoil-NMR: Identification of a Novel Dihydroxy Adamantyl Metabolite

Honrao, Chandrashekhar, Ma, Xiaoyu, Kulkarni, Shashank, Joshi, Vinit, Malamas, Michael, Zvonok, Alexander, Wood, JodiAnne, Strand, David, Guo, Jason J., Makriyannis, Alexandros

Journal:

Frontiers in Pharmacology

Year:

2020

File:

PDF, 1.98 MB

2020

28

Synthesis of Heterocycle-Substituted 1-Aryl-4-piperidones.

Baihua Hu, Michael Malamas, John Ellingboe

Journal:

Year:

2003

File:

PDF, 174 KB

2003

29

Molecular Modeling of the Aldose Reductase-Inhibitor Complex Based on the X-ray Crystal Structure and Studies with Single-Site-Directed Mutants

Singh, Suresh B., Malamas, Michael S., Hohman, Thomas C., Nilakantan, Ramaswamy, Carper, Deborah A., Kitchen, Douglas

Journal:

Journal of Medicinal Chemistry

Year:

2000

Language:

english

File:

PDF, 239 KB

english, 2000

30

Jatrophone, jatrophone derivatives, and analogs. Conformation and reactions with propanethiol

Taylor, Michael D., Smith, Amos B., Malamas, Michael S.

Journal:

Journal of Organic Chemistry

Year:

1983

Language:

english

File:

PDF, 742 KB

english, 1983

31

Novel Benzofuran and Benzothiophene Biphenyls as Inhibitors of Protein Tyrosine Phosphatase 1B with Antihyperglycemic Properties

Malamas, Michael S., Sredy, Janet, Moxham, Christopher, Katz, Alan, Xu, Weixin, McDevitt, Robert, Adebayo, Folake O., Sawicki, Diane R., Seestaller, Laura, Sullivan, Donald

Journal:

Journal of Medicinal Chemistry

Year:

2000

Language:

english

File:

PDF, 1.06 MB

english, 2000

32

Probing the inhibitor-binding site of aldose reductase with site-directed mutagenesis

Thomas C. Hohman, Ossama El-Kabbani, Michael S. Malamas, Kehdih Lai, Tatiana Putilina, Michelle H. McGowan, Yi-Qun Wane, Deborah A. Carper

Journal:

Year:

1998

Language:

english

File:

PDF, 636 KB

english, 1998

33

Synthesis of (-)-bertyadionol

Smith, Amos B., Dorsey, Bruce D., Visnick, Melean., Maeda, Tetsuya., Malamas, Michael S.

Journal:

Journal of the American Chemical Society

Year:

1986

Language:

english

File:

PDF, 409 KB

english, 1986

34

Azole Phenoxy Hydroxyureas as Selective and Orally Active Inhibitors of 5-Lipoxygenase

Malamas, Michael S., Carlson, Richard P., Grimes, David, Howell, Ralph, Glaser, Keith, Gunawan, Iwan, Nelson, James A., Kanzelberger, Mira, Shah, Uresh, Hartman, David A.

Journal:

Journal of Medicinal Chemistry

Year:

1996

Language:

english

File:

PDF, 310 KB

english, 1996

35

Modeling of the outer heliosphere with the realistic solar cycle

Vladislav V. Izmodenov, Yuri G. Malama, Michael S. Ruderman

Journal:

Advances in Space Research

Year:

2008

Language:

english

File:

PDF, 535 KB

english, 2008

36

Facile synthesis of novel spiro[azetidine-2,4′(1′H)-isoquinoline-1′,3′,4(2′H)-triones]

Michael S. Malamas

Journal:

Journal of Heterocyclic Chemistry

Year:

1994

File:

PDF, 288 KB

1994

37

New synthesis of isoxazolidines

Michael S. Malamas, Cynthia L. Palka

Journal:

Journal of Heterocyclic Chemistry

Year:

1996

File:

PDF, 248 KB

1996

38

Quinazolineacetic acids and related analogs as aldose reductase inhibitors

Malamas, Michael S., Millen, Jane

Journal:

Journal of Medicinal Chemistry

Year:

1991

Language:

english

File:

PDF, 1.49 MB

english, 1991

39

Syntheses of tolrestat analogs containing additional substituents in the ring and their evaluation as aldose reductase inhibitors. Identification of potent, orally active 2-fluoro derivatives

Wrobel, Jay, Millen, Jane, Sredy, Janet, Dietrich, Arlene, Gorham, Beverly J., Malamas, Michael, Kelly, Joseph M., Bauman, John G., Harrison, Maria C.

Journal:

Journal of Medicinal Chemistry

Year:

1991

Language:

english

File:

PDF, 2.00 MB

english, 1991

40

Secretion, isotopic labeling and deglycosylation of N-Acylethanolamine acid amidase for biophysical studies

Pavlopoulos, Spiro, Pelekoudas, Dimitrios N., Benchama, Othman, Rawlins, Catherine M., Agar, Jeffrey N., West, Jay M., Malamas, Michael, Zvonok, Nikolai, Makriyannis, Alexandros

Journal:

Protein Expression and Purification

Year:

2017

Language:

english

File:

PDF, 3.04 MB

english, 2017

41

Ruptured ectopic pregnancy: risk factors for a life-threatening condition

Michael Sindos, Athanasia Togia, Theodoros N. Sergentanis, Apostolos Kabagiannis, Fotodotis Malamas, Athanassios Farfaras, Ioannis N. Sergentanis, Vassiliki Bassiotou, Stefanos Antoniou

Journal:

Archives of Gynecology and Obstetrics

Year:

2009

Language:

english

File:

PDF, 181 KB

english, 2009

42

ChemInform Abstract: Antihyperglycemic Activity of New 1,2,4-Oxadiazoline-3,5-diones.

Michael S. Malamas, Janet Sredy, Michael McCaleb, Iwan Gunawan, Brenda Mihan, Donald Sullivan

Journal:

Year:

2001

File:

PDF, 30 KB

2001

43

Aminoimidazoles as Potent and Selective Human β-Secretase (BACE1) Inhibitors

Malamas, Michael S., Erdei, Jim, Gunawan, Iwan, Barnes, Keith, Johnson, Matthew, Hui, Yu, Turner, Jim, Hu, Yun, Wagner, Erik, Fan, Kristi

Journal:

Journal of Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 924 KB

english, 2009

44

Inducibility of liver cytosolic aldehyde dehydrogenase activity in various animal species

Vasilis Vasiliou, Riitta Törrönen, Michael Malamas, Marios Marselos

Journal:

Comparative Biochemistry and Physiology Part C: Comparative Pharmacology

Year:

1989

Language:

english

File:

PDF, 576 KB

english, 1989

45

The Mechanism of Alcohol Intolerance Produced by Various Therapeutic Agents

Vasilis Vasiliou, Michael Malamas, Marios Marselos

Journal:

Basic & Clinical Pharmacology & Toxicology

Year:

1986

Language:

english

File:

PDF, 408 KB

english, 1986

46

ChemInform Abstract: New Oxadiazolidinedione Derivatives as Potent and Selective Human β3 Agonists.

Baihua Hu, Michael Malamas, John Ellingboe, Elwood Largis, Stella Han, Ruth Mulvey, Jeff Tillett

Journal:

Year:

2001

File:

PDF, 32 KB

2001

47

Evaluation of an Estrogen Receptor-β Agonist in Animal Models of Human Disease

Harris, Heather A., Albert, Leo M., Leathurby, Yelena, Malamas, Michael S., Mewshaw, Richard E., Miller, Chris P., Kharode, Yogendra P., Marzolf, James, Komm, Barry S., Winneker, Richard C., Frail, Do

Journal:

Year:

2003

Language:

english

File:

PDF, 337 KB

english, 2003

48

New Azolidinediones as Inhibitors of Protein Tyrosine Phosphatase 1B with Antihyperglycemic Properties

Malamas, Michael S., Sredy, Janet, Gunawan, Iwan, Mihan, Brenda, Sawicki, Diane R., Seestaller, Laura, Sullivan, Donald, Flam, Brenda R.

Journal:

Journal of Medicinal Chemistry

Year:

2000

Language:

english

File:

PDF, 273 KB

english, 2000

49

Estrogen Receptor β Agonism Increases Survival in Experimentally Induced Sepsis and Ameliorates the Genomic Sepsis Signature: A Pharmacogenomic Study

Christaki, Eirini, Opal, Steven M., Keith Jr, James C., Kessinian, Nubar, Palardy, John E., Parejo, Nicolas A., Lavallie, Edward, Racie, Lisa, Mounts, William, Malamas, Michael S., Mewshaw, Richard E.

Journal:

The Journal of Infectious Diseases

Year:

2010

Language:

english

File:

PDF, 5.53 MB

english, 2010

50

Highly Potent, Selective, and Orally Active Phosphodiesterase 10A Inhibitors

Malamas, Michael S., Ni, Yike, Erdei, James, Stange, Hans, Schindler, Rudolf, Lankau, Hans-Joachim, Grunwald, Christian, Fan, Kristi Yi, Parris, Kevin, Langen, Barbara, Egerland, Ute, Hage, Thorsten,

Journal:

Journal of Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 3.22 MB

english, 2011

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